Amide bioisosteres

Amide Bond Bioisosteres: Strategies Synthesis and Successes

pubs.acs.org

To date several amide bioisostere classes are known including 123triazole oxadiazole imidazole tetrazole pyrazole indole pyridine - Information from pubs.acs.org

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Amide bioisosteres information was found here: https://pubs.acs.org/doi/10.1021/acs.jmedchem.0c00530

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Amide Bond Bioisosteres: Strategies Synthesis PubMed

pubmed.ncbi.nlm.nih.gov

The amide functional group plays a key role in the composition of biomolecules including many clinically approved drugs - Information from pubmed.ncbi.nlm.nih.gov

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Amide bioisosteres information was found here: https://pubmed.ncbi.nlm.nih.gov/32686940/

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Ester Bioisosteres Cambridge MedChem Consulting

www.cambridgemedchemconsulting.com

Ester and Amide Bioisosteres Storeoperated calcium entry (SOCE) is a pivotal mechanism in calcium homeostasis bioisosteric replacement of a - Information from www.cambridgemedchemconsulting.com

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Amide bioisosteres information was found here: https://www.cambridgemedchemconsulting.com/resources/bioisoteres/ester_bioisosteres.html

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Application of Amide Bioisosteres in the Optimization of Lead

manu56.magtech.com.cn

Bioisosteres play a role in the same related biochemical system as agonist or antagonist which possessed in related biological activities The amide structure - Information from manu56.magtech.com.cn

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Amide bioisosteres information was found here: http://manu56.magtech.com.cn/progchem/EN/10.7536/PC160414

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Bioisosteres v2 Recent Trends and Tactics Baran Lab

baranlab.org

2018 61 5822 Amide bioisosteres: J Med Chem ASAP General overview: Brown N Bioisosteres in Medicinal Chemistry Wiley‐VCH 2012 - Information from baranlab.org

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Amide bioisosteres information was found here: https://baranlab.org/wp-content/uploads/2020/11/Bioisosteres-v2-Recent-Trends-and-Tactics.pdf

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Amide Bond Bioisosteres: Strategies Synthesis and Successes

experts.nebraska.edu

Herein we review the strategic decisions in selecting an amide bioisostere (the why) synthetic routes to each (the how) and success stories - Information from experts.nebraska.edu

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Amide bioisosteres information was found here: https://experts.nebraska.edu/en/publications/amide-bond-bioisosteres-strategies-synthesis-and-successes

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Isosteres in Medicinal Chemistry

www.scripps.edu

Friedman (1951): Bioisosteres are atoms or molecules that fit Replacement of the sensitive amide bond by various groups - Information from www.scripps.edu

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Amide bioisosteres information was found here: https://www.scripps.edu/baran/images/grpmtgpdf/Mitsos_Feb_06.pdf

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An example of bioisosteres Aminopyrine

labs.chem.ucsb.edu

The trifluoroethylamine can act as an isostere of an amide moiety in peptidebased molecules Trifluoroethylamines as amide isosteres Functional mimicry is - Information from labs.chem.ucsb.edu

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Amide bioisosteres information was found here: https://labs.chem.ucsb.edu/zakarian/armen/10---bioisostere-ucsb-5.potx

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Amide Bond Bioisosteres: Strategies Synthesis and Successes

www.researchgate.net

The amide bond is one of the most important and fascinating functional groups in organic chemistry and biochemistry owing to its widespread occurrence in - Information from www.researchgate.net

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Amide bioisosteres information was found here: https://www.researchgate.net/publication/343091917_Amide_Bond_Bioisosteres_Strategies_Synthesis_and_Successes

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Evaluation of amide bioisosteres leading to 123triazole

www.rti.org

Evaluation of amide bioisosteres leading to 123triazole containing compounds as GPR88 agonists: Design synthesis and structureactivity relationship - Information from www.rti.org

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Amide bioisosteres information was found here: https://www.rti.org/publication/evaluation-amide-bioisosteres-leading-123-triazole-containing-compounds-gpr88-agonists

123Triazoles as Amide Bioisosteres: Discovery of a New Class of

scholarship.miami.edu

123Triazoles as Amide Bioisosteres: Discovery of a New Class of Potent HIV1 Vif Antagonists Idrees Mohammed Indrasena Reddy Kummetha - Information from scholarship.miami.edu

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Amide bioisosteres information was found here: https://scholarship.miami.edu/esploro/outputs/journalArticle/123-Triazoles-as-Amide-Bioisosteres-Discovery-of/991031578297802976

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Amide Bond Bioisosteres: Strategies Synthesis and Successes

europepmc.org

Amide Bond Bioisosteres: Strategies Synthesis and Successes Herein we review the strategic decisions in selecting an amide bioisostere (the why) - Information from europepmc.org

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Amide bioisosteres information was found here: https://europepmc.org/article/med/32686940

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Evaluation of 123‐Triazoles as Amide Bioisosteres In Cystic

chemistry-europe.onlinelibrary.wiley.com

Abstract The 123triazole has been successfully utilized as an amide bioisostere in multiple therapeutic contexts - Information from chemistry-europe.onlinelibrary.wiley.com

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Amide bioisosteres information was found here: https://chemistry-europe.onlinelibrary.wiley.com/doi/10.1002/chem.201805919

Reductive Functionalization of Amides in Synthesis and for

www.frontiersin.org

Reductive functionalization of amides in context of latestage functionalization and bioisosteres (A) Comparison of triflic - Information from www.frontiersin.org

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Amide bioisosteres information was found here: https://www.frontiersin.org/articles/655849

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Bioisostere Wikipedia

en.wikipedia.org

In medicinal chemistry bioisosteres are chemical substituents or groups with similar Procainamide an amide has a longer duration of action than Procaine - Information from en.wikipedia.org

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Amide bioisosteres information was found here: https://en.wikipedia.org/wiki/Bioisostere

Application of Bioisosteres in Drug Design

www.f.u-tokyo.ac.jp

~Amide and Ester Isosteres ~Phenyl Ring Isosteres 3 Oxetanes in Drug Discovery ~Physicochemical Properties of Oxetanes - Information from www.f.u-tokyo.ac.jp

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Amide bioisosteres information was found here: https://www.f.u-tokyo.ac.jp/~kanai/seminar/pdf/Lit_Y_Morita_M1.pdf

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14Disubstituted 123Triazoles as Amide Bond Surrogates

www.mdpi.com

This study shows that the 123triazole is not in all cases a universal bioisostere for a transamide bond as their incorporation into the peptide can - Information from www.mdpi.com

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Amide bioisosteres information was found here: https://www.mdpi.com/1420-3049/25/16/3576/htm

SwissBioisostere 2021: updated structural Oxford Academic

academic.oup.com

At several stages of drug discovery bioisosteric replacement is a common (26) can arguably be considered as true amide bioisosteres - Information from academic.oup.com

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Amide bioisosteres information was found here: https://academic.oup.com/nar/advance-article/doi/10.1093/nar/gkab1047/6426059

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Trisubstituted acylhydrazines as tertiary amide bioisosteres: HCV

www.infona.pl

The use of a trisubstituted acylhydrazine as an isostere of a tertiary amide was explored in a series of HCV NS5B thumb site II inhibitors - Information from www.infona.pl

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Amide bioisosteres information was found here: https://www.infona.pl/resource/bwmeta1.element.elsevier-4ae2566f-afdd-3894-ba3d-a0f5fa8dd36e

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Identification of amide bioisosteres of triazole oxytocin

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A series of amides were investigated as potential bioisosteres of previously reported triazole oxytocin antagonists although SAR for potency and - Information from www.semanticscholar.org

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Amide bioisosteres information was found here: https://www.semanticscholar.org/paper/Identification-of-amide-bioisosteres-of-triazole-Brown-Ellis/b4e27e118755b4cb97c85a87bedd2e527d23959b

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Stable pantothenamide bioisosteres the journal of antibiotics

www.nature.com

Stable pantothenamide bioisosteres: novel antibiotics for Grampositive bacteria Patrick A M Jansen Danique A van der Krieken - Information from www.nature.com

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Amide bioisosteres information was found here: https://www.nature.com/articles/s41429-019-0196-6

Bioisosterism: A Rational Approach in Drug Design

mch.estranky.sk

Amide Group Bioisosteres successful use of bioisosteres have been included the isosterism is that bioisosteres affect the same phar - Information from mch.estranky.sk

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Amide bioisosteres information was found here: https://mch.estranky.sk/file/228/1996chemrev96-3147-76_bioisosterism.pdf

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Applications of fluorine to the construction of bioisosteric

www.tandfonline.com

In addition the classic exploitation of trifluoroethylamine group as an amide bioisostere is discussed In each of the case studies presented - Information from www.tandfonline.com

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Amide bioisosteres information was found here: https://www.tandfonline.com/doi/abs/10.1080/17460441.2021.1933427

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Allenamide as a bioisostere of acrylamide in the design and

pubs.rsc.org

Our study indicates that the allenamide group could serve as an alternative electrophilic warhead in the design of targeted covalent inhibitors and this - Information from pubs.rsc.org

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Amide bioisosteres information was found here: https://pubs.rsc.org/en/content/articlelanding/2018/md/c7md00571g

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123triazoles as amide bioisosteres: Discovery of a new class of

miami.pure.elsevier.com

123triazoles as amide bioisosteres: Discovery of a new class of potent HIV1 Vif antagonists Idrees Mohammed Indrasena Reddy Kummetha - Information from miami.pure.elsevier.com

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Amide bioisosteres information was found here: https://miami.pure.elsevier.com/en/publications/123-triazoles-as-amide-bioisosteres-discovery-of-a-new-class-of-p

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The Influence of Bioisosteres in Drug Design SpringerLink

link.springer.com

The application of bioisosteres in drug discovery is a establish an interaction with the C atom of the backbone amide CO of Asn98 at a - Information from link.springer.com

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Amide bioisosteres information was found here: https://link.springer.com/chapter/10.1007/7355_2013_29

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Amide bioisosteres Publications PubFacts

www.pubfacts.com

College of Pharmacy Yeungnam University Gyeongsan 38541 Korea Two novel bioisosteres of cabozantinib and were designed and synthesized The benzene ring - Information from www.pubfacts.com

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Amide bioisosteres information was found here: https://www.pubfacts.com/search/Amide+bioisosteres

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Drug design principles Stereoelectronics

www.stereoelectronics.org

The role of the common functional groups Isosteres and bioisosteres and secondary amines could be used to check whether the amide is acting as an HBD - Information from www.stereoelectronics.org

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Amide bioisosteres information was found here: https://www.stereoelectronics.org/webDD/DD_04.html

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3MF5: Hepatitis C virus polymerase NS5B (BK) with amide

www.rcsb.org

Conformational modeling has been successfully applied to the design of cyclic bioisosteres used to replace a conformationally rigid amide - Information from www.rcsb.org

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Amide bioisosteres information was found here: https://www.rcsb.org/structure/3MF5

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Trisubstituted acylhydrazines as tertiary amide bioisosteres

agris.fao.org

Trisubstituted acylhydrazines as tertiary amide bioisosteres: HCV NS5B polymerase inhibitors [2012] Canales Eda Carlson Joseph S Appleby Todd - Information from agris.fao.org

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Amide bioisosteres information was found here: https://agris.fao.org/agris-search/search.do?recordID=US201500130803

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PRIME PubMed Identification of amide bioisosteres of triazole

www.unboundmedicine.com

A series of amides were investigated as potential bioisosteres of previously reported triazole oxytocin antagonists A range of potent analogues were - Information from www.unboundmedicine.com

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Amide bioisosteres information was found here: https://www.unboundmedicine.com/medline/citation/20189387/Identification_of_amide_bioisosteres_of_triazole_oxytocin_antagonists_

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Chemical Biology and Drug Development Rana Lab

ranalab.ucsd.edu

(2016) 123Triazoles as amide bioisosteres: Discovery of a new class of potent HIV1 Vif antagonists Journal of Medicinal Chemistry 59 76777682 - Information from ranalab.ucsd.edu

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Amide bioisosteres information was found here: https://ranalab.ucsd.edu/sample-page/chemical-biology-and-drug-development/

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Surveying heterocycles as amide bioisosteres within a series

www.meta.org

Surveying heterocycles as amide bioisosteres within a series of mGlu7 NAMs: Discovery of VU6019278 Bioorganic & Medicinal Chemistry Letters - Information from www.meta.org

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Amide bioisosteres information was found here: https://www.meta.org/papers/surveying-heterocycles-as-amide-bioisosteres/30910459

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Design and Synthesis of Bioisosteres of Acylhydrazones as

research.rug.nl

The most successful bioisostere is equipotent bears an amide linker and we confirmed its binding mode by Xray crystallography Having some validated - Information from research.rug.nl

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Amide bioisosteres information was found here: https://research.rug.nl/files/76824714/Jumde_et_al_2018_ChemMedChem.pdf

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Jake Doiron School of Graduate Studies LSU Health New

graduatestudies.lsuhsc.edu

Structural Consequences of the 123Triazole as an Amide Bioisostere in Evaluation of 123triazoles as amide bioisosteres in cystic fibrosis - Information from graduatestudies.lsuhsc.edu

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Amide bioisosteres information was found here: https://graduatestudies.lsuhsc.edu/md_phd/jake_doiron.aspx

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Amide Bond Bioisosteres: Strategies Synthesis and Successes

www.x-mol.com

The amide functional group plays a key role in the composition of biomolecules including many clinically approved drugs - Information from www.x-mol.com

Information accuracy 100%
Amide bioisosteres information was found here: https://www.x-mol.com/paper/1285278876615491584

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Optimizing Drug Properties LeadtoDrug Design UZH

www.chem.uzh.ch

Blocks hydrolysis of terminal amide Metabolic Drug Stability Replace labile ester with more stable urethane or amide bioisostere for amide - Information from www.chem.uzh.ch

Information accuracy 100%
Amide bioisosteres information was found here: http://www.chem.uzh.ch/zerbe/MedChem/MedChem5_Lead.pdf

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15Disubstituted 123Triazoles as Amide Bond Isosteres

hal.archives-ouvertes.fr

bioisosteres of amide bonds in peptidomimetics to modify the pharmacological properties of peptides or proteins1620 The systematic - Information from hal.archives-ouvertes.fr

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Amide bioisosteres information was found here: https://hal.archives-ouvertes.fr/hal-03178434/document

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Preparation of novel anthranilic acids as antibacterial agents

www.sigmaaldrich.com

Extensive evaluation of alternative amide bioisosteres connecting the A and the Brings by Atli Thorarensen Brian D Wakefield Donna L Romero - Information from www.sigmaaldrich.com

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Amide bioisosteres information was found here: https://www.sigmaaldrich.com/FR/fr/tech-docs/paper/84632

Bioisosterism: A Useful Strategy for Molecular Modification

www.lassbio.icb.ufrj.br

Other common examples of amide function bioisosteres include the “retroamide” groups ie: ACONHB ⇒ A NHCOB and alkylydene (CHCH2) [472] Wrobel and - Information from www.lassbio.icb.ufrj.br

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Amide bioisosteres information was found here: http://www.lassbio.icb.ufrj.br/download/cursos_semin/2015/bioisosterism2015.pdf

The Use of Bioisosterism in Drug Design and Molecular

citeseerx.ist.psu.edu

Bioisosteres are atoms or group of molecules that fit the broadest definition for isosteres They Amide group bioisosteres 22 B4 - Information from citeseerx.ist.psu.edu

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Amide bioisosteres information was found here: http://citeseerx.ist.psu.edu/viewdoc/download?doi=10.1.1.301.520&rep=rep1&type=pdf

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PBDA 1 Lecture 15 Bioisosterism analogs Flashcards Quizlet

quizlet.com

Isosteric replacemet or Bioisosteric replacement Replacement or modification of specific Image: Nonclassical bioisosteres for Amide group - Information from quizlet.com

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Amide bioisosteres information was found here: https://quizlet.com/431936539/pbda-1-lecture-15-bioisosterism-analogs-flash-cards/

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Amide Bond Bioisosteres: Strategies Synthesis 文献云下载

download.xuebalib.com

bioisosteres in drug design2731 along with a more recent review focused on amide bioisosteres32 This perspective aims to be a reference - Information from download.xuebalib.com

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Amide bioisosteres information was found here: http://download.xuebalib.com/ba3rRqG0nbWr.pdf

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Bioisosteric Replacement as a Tool in AntiHIV Drug Design

mdpi-res.com

Figure 7 Diaminosquarate bioisostere for the guanidine moiety as a novel HIV1 TatTAR RNA inhibitor Amide and Ester Bioisosterism - Information from mdpi-res.com

Information accuracy 100%
Amide bioisosteres information was found here: https://mdpi-res.com/d_attachment/pharmaceuticals/pharmaceuticals-13-00036/article_deploy/pharmaceuticals-13-00036-v2.pdf

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Pyrazoles as nonclassical bioisosteres in DOCKSCICOM

docksci.com

The results indicate that pyrazoles are suitable bioisosteric replacements of amide functional groups The study is an example of managing bioisosteric - Information from docksci.com

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Amide bioisosteres information was found here: https://docksci.com/pyrazoles-as-non-classical-bioisosteres-in-prolylcarboxypeptidase-prcp-inhibitor_5af52d96d64ab26364f70562.html

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bioisosterismopdf UFPR

www.quimica.ufpr.br

Bioisosteres are atoms or group of molecules that fit the broadest definition for isosteres They Amide group bioisosteres 22 B4 - Information from www.quimica.ufpr.br

Information accuracy 100%
Amide bioisosteres information was found here: http://www.quimica.ufpr.br/nunesgg/QIM__PG/material%20para%20estudo/bioisosterismo.pdf

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12Difunctionalized Bicyclo[111]pentanes ChemRxiv

chemrxiv.org

Bioisosteres for ortho/metaSubstituted Arenes and 21 underwent amide bond coupling to obtain Meclizine bioisosteres 18 and 19 in 45% and - Information from chemrxiv.org

Information accuracy 100%
Amide bioisosteres information was found here: https://chemrxiv.org/engage/api-gateway/chemrxiv/assets/orp/resource/item/60c7511fbb8c1a389e3dbc11/original/1-2-difunctionalized-bicyclo-1-1-1-pentanes-long-sought-after-bioisosteres-for-ortho-meta-substituted-arenes.pdf

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Stephen Aller (0000000303795534) ORCID

orcid.org

Structural Consequences of the 123‐Triazole as an Amide Bioisostere in Analogues of the Cystic Fibrosis Drugs VX‐809 and VX‐770 - Information from orcid.org

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Amide bioisosteres information was found here: https://orcid.org/0000-0003-0379-5534

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Design and Synthesis of Phosphonoacetic Acid (PPA) Ester

journals.sagepub.com

Design and Synthesis of Phosphonoacetic Acid (PPA) Ester and Amide in order to verify the possible interaction of the proposed bioisosteric moieties - Information from journals.sagepub.com

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Amide bioisosteres information was found here: https://journals.sagepub.com/doi/abs/10.1177/095632020301400403

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ChemMedChem on Twitter: "K Auclair McGillU K Saliba

twitter.com

et al report triazole rings as amide #bioisosteres Such #antimalarial pantothenamide analogues resist degradation by pantetheinases - Information from twitter.com

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Amide bioisosteres information was found here: https://twitter.com/chemmedchem/status/1068401291460820992

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Mark Turlington Berry College

www.berry.edu

Evaluation of 123Triazoles as Amide Bioisosteres in Cystic Fibrosis Transmembrane Conductance Regulator Modulators VX770 and VX809 Chem Eur J 2019 - Information from www.berry.edu

Information accuracy 100%
Amide bioisosteres information was found here: https://www.berry.edu/academics/fs/_assets/mturlington-cv.pdf

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Oxetanes SpiroChem TailorMade Molecules

spirochem.com

Oxetanylamines can be seen and used as bioisosteres of amide fragments Why oxetanes? The use of oxetanes in drug discovery has known an - Information from spirochem.com

Information accuracy 100%
Amide bioisosteres information was found here: https://spirochem.com/catalog/oxetanes.html

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In vitro evaluation of Nmethyl amide tripeptidomimetics as

pharmacy.ku.dk

The aim of the present study was to evaluate the general application of Nmethyl amide bioisosteres as peptide bond replacements in tripeptides in order to - Information from pharmacy.ku.dk

Information accuracy 100%
Amide bioisosteres information was found here: https://pharmacy.ku.dk/research/cns-drug-delivery-barrier-modelling/?pure=en%2Fpublications%2Fin-vitro-evaluation-of-nmethyl-amide-tripeptidomimetics-as-substrates-for-the-human-intestinal-ditripeptide-transporter-hpept1(f644a89d-f856-4808-9db0-1cbb633a717a).html

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Publications Dr James A Bull Imperial College London

www.imperial.ac.uk

title {Aminooxetanes as amide isosteres by an alternative AB Bioisosteres provide valuable design elements for medicinal chemists to adjust the - Information from www.imperial.ac.uk

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Amide bioisosteres information was found here: https://www.imperial.ac.uk/people/j.bull/publications.html?respub-action=citation.html&id=1234377&noscript=noscript

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The powerful symbiosis between synthetic and medicinal

www.future-science.com

Bioisosteres have similar shape and connectivity to the Although conformational studies of an Ntrifluoromethyl amide showed a lower - Information from www.future-science.com

Information accuracy 100%
Amide bioisosteres information was found here: https://www.future-science.com/doi/pdf/10.4155/fmc-2021-0062

PDB 4eo8 citation summary ‹ Protein Data Bank in Europe

www.ebi.ac.uk

4eo8: Trisubstituted acylhydrazines as tertiary amide bioisosteres: HCV NS5B polymerase inhibitors - Information from www.ebi.ac.uk

Information accuracy 100%
Amide bioisosteres information was found here: https://www.ebi.ac.uk/pdbe/entry/pdb/4eo8/citations

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Article Structureactivity relationships of antiplasmodial

escholarship.mcgill.ca

We previously reported that replacement of the labile amide bond with a triazole ring not amide bioisosteres · Plasmodium falciparum - Information from escholarship.mcgill.ca

Information accuracy 100%
Amide bioisosteres information was found here: https://escholarship.mcgill.ca/concern/articles/dv13zz06x

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LEMOINE SAMUEL J MS The Development and Uncg

libres.uncg.edu

Bioisosteric Software Program for the Development of New Pharmaceuticals (2014) Parent compound with amidebased bioisosteres and - Information from libres.uncg.edu

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Amide bioisosteres information was found here: https://libres.uncg.edu/ir/uncg/f/Lemoine_uncg_0154M_11438.pdf

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Search results Scholarly Publications

scholarlypublications.universiteitleiden.nl

Enabled Filters () Amide bioisosteres Sort Options Date (year) · Author / Creator · Title Refine Results Availability Open access (1) + Faculty - Information from scholarlypublications.universiteitleiden.nl

Information accuracy 100%
Amide bioisosteres information was found here: https://scholarlypublications.universiteitleiden.nl/search?type=dismax&f%5B0%5D=mods_subject_topic_ms%3AAmide%5C%20bioisosteres

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Application of Amide Bioisosteres in the JGlobal

jglobal.jst.go.jp

Article “Application of Amide Bioisosteres in the Optimization of Lead Compounds” Detailed information of the JGLOBAL is a service based on - Information from jglobal.jst.go.jp

Information accuracy 100%
Amide bioisosteres information was found here: http://jglobal.jst.go.jp/en/public/20090422/201702270917809656

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Surveying heterocycles as amide bioisosteres within a series of

www.researcher-app.com

as bioisosteric replacements for a metabolically labile amide moiety within a 134oxadizaole ring system as an effective bioisostere for the amide - Information from www.researcher-app.com

Information accuracy 100%
Amide bioisosteres information was found here: https://www.researcher-app.com/paper/2476633

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Amidinohydrazones as Guanidine Bioisosteres BetaSheetorg

beta-sheet.org

Abstract╨We describe a new class of potent nonamidebased small molecule thrombin inhibitors in which an amidinohydrazone - Information from beta-sheet.org

Information accuracy 100%
Amide bioisosteres information was found here: http://beta-sheet.org/resources/86-Aminohydrazones-as-Guanidine.pdf

Advances in Triazole Chemistry Page 46 Google Books Result

books.google.com

4Hydroxy123triazole moiety as bioisostere of the carboxylic acid function: a Evaluation of 123‐triazoles as amide bioisosteres in cystic fibrosis - Information from books.google.com

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Bioisosteres Hiroyuki Kobayashi Jan SlidePlayer

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An example of bioisosteres Aminopyrine Marketed as an analgesic and Amide isosteres have typically been of interest as a means of modulating polarity - Information from slideplayer.com

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The Dopamine Receptors Page 108 Google Books Result

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59 Binding affinities of several amides with butylene linkers Ki values in nM As described for DPATs heterocyclic bioisosteres are also known for the - Information from books.google.com

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Current Medicinal Chemistry Page 384 Google Books Result

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COR Scheme XllI: Synthesis of 2monosubstituted amide bioisosteres of pseudoglycerides Reagents and conditions: a) RiCOCl diethylether: or a) - Information from books.google.com

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(2012 Jul 18) Gilead Sciences Inc Foster City: Trisubstituted acylhydrazines as tertiary amide bioisosteres: HCV NS5B polymerase inhibitors By a News - Information from books.google.com

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A triazole ring and a ketopiperazine moiety were introduced as bioisosteres of the amide to improve the instability of the peptides [55] - Information from books.google.com

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New Developments in Medicinal Chemistry

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Subsequently the authors synthesized amide bioisosteres of the previously antagonists and the higher synthetic accessibility of the amides (Fig - Information from books.google.com

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Bioisosteres in Medicinal Chemistry Page 38 Google Books Result

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These compounds exemplify the problems outlined above with two amide groups and a sulfonamide (plus a carboxylic acid) Molecular modeling indicated that - Information from books.google.com

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Microbial proteasomes as drug targets PLOS

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In order to improve the pharmacokinetic properties of DPLG2 the Cterminal amide was replaced with its bioisosteres phenylimidazole [45] - Information from journals.plos.org

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Publications The Knowles Group

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Understanding Chemoselectivity in ProtonCoupled Electron Transfer: A Kinetic Study of Amide and Thiol Activation Guanqi Qiu Robert R Knowles - Information from knowleslab.princeton.edu

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Pharmacokinetics in Modern Drug Design Medicinal Chemistry

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Esters and amides are major groups of carrierlinked prodrugs Bioisosteres also allow for the development of “metoo” drugs - Information from pharmafactz.com

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[65] 20 was reacted with DSG to install an amidelinked alkyl linker The product 21 was then reacted with the E3binding pentapeptide sequence to displace - Information from www.explorationpub.com

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Amide: Definition Structure & Formation Studycom

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In chemistry amides are compounds that contain nitrogen atoms Learn more about the definition structure and formation of amides - Information from study.com

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Amines and Amides Chemistry for Majors Lumen Learning

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Amines are molecules that contain carbonnitrogen bonds The nitrogen atom in an amine has a lone pair of electrons and three bonds to other atoms - Information from courses.lumenlearning.com

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Preparation of amides using DCC (video) Khan Academy

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Amide Biochemistry Flashcards Draw it to Know it

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Amide Functional Group • The nitrogen variant of an ester A C bonded to a hydrogen doublebonded to an O singlebonded to an N which is also bound to - Information from www.drawittoknowit.com

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Amide bioisosteres

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EDUCATION Amide Bond Bioisosteres: Strategies Synthesis PubMed

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EDUCATION Amide Bond Bioisosteres: Strategies Synthesis and Successes

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EDUCATION An example of bioisosteres Aminopyrine

EDUCATION Amide Bond Bioisosteres: Strategies Synthesis and Successes

EDUCATION Evaluation of amide bioisosteres leading to 123triazole

EDUCATION 123Triazoles as Amide Bioisosteres: Discovery of a New Class of

EDUCATION Amide Bond Bioisosteres: Strategies Synthesis and Successes

EDUCATION Evaluation of 123‐Triazoles as Amide Bioisosteres In Cystic

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EDUCATION Application of Bioisosteres in Drug Design

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EDUCATION Trisubstituted acylhydrazines as tertiary amide bioisosteres: HCV

EDUCATION Identification of amide bioisosteres of triazole oxytocin

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EDUCATION Bioisosterism: A Rational Approach in Drug Design

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EDUCATION The Influence of Bioisosteres in Drug Design SpringerLink

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EDUCATION Amide Bond Bioisosteres: Strategies Synthesis and Successes

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EDUCATION The powerful symbiosis between synthetic and medicinal

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EDUCATION Application of Amide Bioisosteres in the JGlobal

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EDUCATION The Dopamine Receptors Page 108 Google Books Result

EDUCATION Current Medicinal Chemistry Page 384 Google Books Result

EDUCATION Issues in Medical Chemistry: 2013 Edition

EDUCATION DiversityOriented Synthesis: Basics and Applications in

EDUCATION New Developments in Medicinal Chemistry

EDUCATION Bioisosteres in Medicinal Chemistry Page 38 Google Books Result

EDUCATION Microbial proteasomes as drug targets PLOS

EDUCATION Publications The Knowles Group

EDUCATION Pharmacokinetics in Modern Drug Design Medicinal Chemistry

EDUCATION AMIDE: a Medical Image Data Analysis Tool

EDUCATION Current strategies for the design of PROTAC linkers: a critical

EDUCATION Amide: Definition Structure & Formation Studycom

EDUCATION Properties of Amides YouTube

EDUCATION Amines and Amides Chemistry for Majors Lumen Learning

EDUCATION Preparation of amides using DCC (video) Khan Academy

Amide Bond Bioisosteres: Strategies Synthesis and Successes

Amide Bond Bioisosteres: Strategies Synthesis PubMed

Ester Bioisosteres Cambridge MedChem Consulting

Application of Amide Bioisosteres in the Optimization of Lead

Bioisosteres v2 Recent Trends and Tactics Baran Lab

Amide Bond Bioisosteres: Strategies Synthesis and Successes

Isosteres in Medicinal Chemistry

An example of bioisosteres Aminopyrine

Amide Bond Bioisosteres: Strategies Synthesis and Successes

Evaluation of amide bioisosteres leading to 123triazole

123Triazoles as Amide Bioisosteres: Discovery of a New Class of

Amide Bond Bioisosteres: Strategies Synthesis and Successes

Evaluation of 123‐Triazoles as Amide Bioisosteres In Cystic

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Bioisostere Wikipedia

Application of Bioisosteres in Drug Design

14Disubstituted 123Triazoles as Amide Bond Surrogates

SwissBioisostere 2021: updated structural Oxford Academic

Trisubstituted acylhydrazines as tertiary amide bioisosteres: HCV

Identification of amide bioisosteres of triazole oxytocin

Stable pantothenamide bioisosteres the journal of antibiotics

Bioisosterism: A Rational Approach in Drug Design

Applications of fluorine to the construction of bioisosteric

Allenamide as a bioisostere of acrylamide in the design and

123triazoles as amide bioisosteres: Discovery of a new class of

The Influence of Bioisosteres in Drug Design SpringerLink

Amide bioisosteres Publications PubFacts

Drug design principles Stereoelectronics

3MF5: Hepatitis C virus polymerase NS5B (BK) with amide

Trisubstituted acylhydrazines as tertiary amide bioisosteres

PRIME PubMed Identification of amide bioisosteres of triazole

Chemical Biology and Drug Development Rana Lab

Surveying heterocycles as amide bioisosteres within a series

Design and Synthesis of Bioisosteres of Acylhydrazones as

Jake Doiron School of Graduate Studies LSU Health New

Amide Bond Bioisosteres: Strategies Synthesis and Successes

Optimizing Drug Properties LeadtoDrug Design UZH

15Disubstituted 123Triazoles as Amide Bond Isosteres

Preparation of novel anthranilic acids as antibacterial agents

Bioisosterism: A Useful Strategy for Molecular Modification

The Use of Bioisosterism in Drug Design and Molecular

PBDA 1 Lecture 15 Bioisosterism analogs Flashcards Quizlet

Amide Bond Bioisosteres: Strategies Synthesis 文献云下载

Bioisosteric Replacement as a Tool in AntiHIV Drug Design

Pyrazoles as nonclassical bioisosteres in DOCKSCICOM

bioisosterismopdf UFPR

12Difunctionalized Bicyclo[111]pentanes ChemRxiv

Stephen Aller (0000000303795534) ORCID

Design and Synthesis of Phosphonoacetic Acid (PPA) Ester

ChemMedChem on Twitter: "K Auclair McGillU K Saliba

Mark Turlington Berry College

Oxetanes SpiroChem TailorMade Molecules

In vitro evaluation of Nmethyl amide tripeptidomimetics as

Publications Dr James A Bull Imperial College London

The powerful symbiosis between synthetic and medicinal

PDB 4eo8 citation summary ‹ Protein Data Bank in Europe

Article Structureactivity relationships of antiplasmodial

LEMOINE SAMUEL J MS The Development and Uncg

Search results Scholarly Publications

Application of Amide Bioisosteres in the JGlobal

Surveying heterocycles as amide bioisosteres within a series of

Amidinohydrazones as Guanidine Bioisosteres BetaSheetorg

Advances in Triazole Chemistry Page 46 Google Books Result

Bioisosteres Hiroyuki Kobayashi Jan SlidePlayer

The Dopamine Receptors Page 108 Google Books Result

Current Medicinal Chemistry Page 384 Google Books Result

Issues in Medical Chemistry: 2013 Edition

DiversityOriented Synthesis: Basics and Applications in

New Developments in Medicinal Chemistry

Bioisosteres in Medicinal Chemistry Page 38 Google Books Result

Microbial proteasomes as drug targets PLOS

Publications The Knowles Group

Pharmacokinetics in Modern Drug Design Medicinal Chemistry

AMIDE: a Medical Image Data Analysis Tool

Current strategies for the design of PROTAC linkers: a critical

Amide: Definition Structure & Formation Studycom

Properties of Amides YouTube

Amines and Amides Chemistry for Majors Lumen Learning

Preparation of amides using DCC (video) Khan Academy

Amide Biochemistry Flashcards Draw it to Know it